肿瘤已经成为威胁人类生命的一大杀手，人类健康成为了世界难题，那么有没有什么能够抵抗肿瘤的药物呢？武汉贝尔卡为大家统计较为常见的抗肿瘤类原料药及中间体，以及其他种类的原料药和中间体的汇总！
抗肿瘤类原料药及中间体
PRODUCTSPECIFICATION
★原料药
卡铂CarboplatinEP/USP/CP
顺铂CisplatinEP/USP/CP
奥沙利铂OxaliplatinEP5
奈达铂NedaplatinIn-House
依铂EptaplatinIn-House
吉西他滨GemcitabineIn-House
卡培他滨CapecitabineIn-House
替氟TegafurCP/JP
吉莫斯特GimeracilIn-House
氧嗪酸钾OteracilpotassiumIn-House
培美曲塞二钠PemetrexedDisodiumIn-House
唑来膦酸ZoledronicAcidIn-House
异环膦酸铵IfosfamideUSP/CP
氯法拉滨ClofarabineIn-House
★中间体
①铂系列药物中间体
氯亚铂酸钾
Potassiumtetrachloroplatinate(I) [10025-99-7]
二碘二氨合铂
Diododiammineplatinum
二硝基环己二胺铂
DACHPL ATINUMDINITRATE
顺式-二氯~[反式-(-)-1 , 2-环己二胺]铂
Cis-dichloro(trans 1-1,2-cyclohexanediamine ) pt(I)
左旋-反式-1 , 2-环己二胺
( 1R,2R ) -(-)-1,2-diaminocyclohexane[20439-47-8]
反式-1,2-环己二胺
Trans-1 , 2-diaminocyclohexane[1121-22-8]
环丁基甲酸
Cyclobutanecarboxylicacid[3721-95-7]
②卡培他滨中间体intermediateofCapecitabine
三乙酰基-5-脱氧核糖Assay298.5%
1 , 2 , 3-triacetyl-5-deoxy- B- D-Ribose[62211-93-2]
③吉西他滨中间体IntermediatesofGemcitabine
双丙醇-D-甘露糖醇; 1,2:5,6-1 -异亚丙基-D-mannitolAssay≥95%
1,2:5,6- Bis-O-(1-methylethylidene)-D-mannitol[1707-77-3]
2-脱氧-2 , 2-氟戊呋喃糖1-酮-3 , 5-=按息香酸盐(又名核酮糖) Assay295%
2-Deoxy-2,2-difluoro-D-erythro-pentofuranos-1-ulose-3,5-dibenzoate[122111-01-7]
④培美曲塞二钠中间体IntermediatesofPemetrexedDisodium
培美曲塞酸Pemetrexed[137281-23-3]
N-(4-[2-(2-氨基-4, 7-=氢-4氧1H-吡咯[2 , 3-D]嘧啶-5-基)
乙基]苯甲酰)-L-谷氨酸= Z酯对甲苯磺酸盐
(N-[4-[2-(2-amino-4,7-dihydro-4-oxo-3H-pyrrolo[2,3-d]
pyrimidin-5-yl)ethyl]benzoyI]L -Glutamicacid[165049-28-5]
4-[2-(2-氨基-4, 7-=氢-4-氧1H-吡咯[2,3-D-]嘧啶- 5-基)Z基]苯甲酸
4-[2-(2-amino-4-oxo-4,7-dihydro-4-oxo-3H-pyrrolo(2,3-d)
pyrimidin-5-yl)ethyl]benzoicacid[137281 -39-1]
⑤异环磷酰胺中间体Intermediateoflfosfamide
3-(2-氯乙酰基)-2-[(2-氯Z基)氨基]四氢2H-1 , 3 , 2-恶磷2-氧化物
Ifosfamideacylationobjects[72578-71-3]
⑥氯法拉滨中间体IntermediatesofClofarabine
2,3,5-三苯甲酰基_B-D-呋喃核糖
beta-D-Ribofuranose2,3,5-tribenzoate[67525-66-0]
1,3,5-1 =-O苯甲酰基2-脱氧- 2-氟alpha-L-阿拉伯呋喃糖
1,3,5-Tri-O-benzoyl-2-deoxy-2-fluoro-alpha-L-arabinofuranosev[171721-00-9]
抗真菌类原料药及中间体
PRODUCTSPECIFICATION
★原料药
盐酸特比萘芬TerbinafineHydrochlorideEP5.3
盐酸布替萘芬ButenafineHydrochlorideIn-House
伏立康唑VoriconazoleIn-House
★盐酸特比萘芬中间体IntermediatesofTerbinafineHydrochloride
N-甲基- 1-萘甲胺
N-methyl-1-naphthalenemethylamine[14489-75-9]
3,3-二甲基-1-丁炔
3 , 3-Dimethyl-1-Butyne[917-92-0]
反式-1,3-二氯丙烯
Trans- 1,3-dichloropropene[10061-02-6]
1-氯-6, 6-二甲基-2-庚烯-4-炔
1-chloro-6,6- dimethyl-2-heptyene-4-alkyne[126764-17-8]
特比萘芬碱基
Terbinafinebase
抗高血压类原料药及中间体
PRODUCTSPECIFICATION
★原料药
尼嗦地平NisoldipineIn-House
醌地平CilnidipineIn-House
盐酸马尼地平ManidipinedihydrochlorideIn-House
非洛地平FelodipineUSP30
托拉塞米TorasemideUSP30
盐酸雷诺嗪RanolazinedihydrochlorideIn-House
★中间体
①西尼地平中间体IntermediateofCilnidipine
3-氨基-2-丁烯酸肉桂酯
3-AminoCrotonicAcidCinnamylEster
②托拉塞米中间体IntermediateofTorasemide
[4-(3-甲基苯基)氨基]吡啶- 3-磺酰胺
[4-(3-Methylpheny)amino]pyridine-3-sulphonamide[72811-73-5]
镇痛麻醉类原料药及中间体
PRODUCTSPECIFICATION
★原料药
罗哌卡因盐酸盐
RopivacaineHydrochlorideUSP
罗哌卡因甲磺酸盐
RopivacaineMesilateIn-House .
布比卡因盐酸盐
BupivacaineHydrochlorideUSP/EP
S-布比卡因盐酸盐
LevobupivacaineHydrochloride
顺苯磺阿曲库铵
CisatracuriumBesylateIn-House
苯磺酸阿曲库铵
AtracuriumbesylateUSP/EP
★中间体
①卡因类中间体IntermediatesofAnalgesiaanaesthesia
(S)-N-(2,6-- = 甲苯基)- 2-哌啶酰胺
(S)-N-(2,6-dimethylpheny)-piperidine- 2-carboxylicamide[27262-40-4]
N-(2,6-二甲苯基)-2-哌啶酰胺
N-(2,6-dimethylpheny)-piperidine- 2-carboxylicamide[15883-20-2]
②顺苯磺阿曲库铵类中间体IntermediatesofCisatracuriumbesylate
R-s四氢罂粟碱-N-乙酰-L-亮氨酸
R-tetrahydropapaverine-N-acetyl-L-leucinate[141109-12-8]
R-四氢罂粟碱盐酸盐
(R)-tetrahydropapaverinehydrochloride[54417-53-7]
其他类原料药及中间体
PRODUCTSPECIFICATION
★原料药
米格列奈钙
MitiglinidecalciumIn-House
消旋卡够曲
RacecadotrilEP6.2
氨芬酸钠
AmfenacesodiumIn-House
★中间体
①米格列奈钙中间体IntermediatesofMitiglinidecalcium
S-苄基琥珀酸
S- Benzylsuccinincacid[3972-36-9]
顺式全氢异吲哚
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